1: 96 percent / AcOH / xylene / 6.5 h / Heating 2: 1.) NaH / 1.) DMF, RT, 0.5 h, 2.) DMF, RT, 1 h 3: 68 percent / Bu3SnN3 / xylene / 88 h / Heating View Scheme
参考文献
Bernhart, Claude A.; Perreaut, Pierre M.; Ferrari, Bernard P.; Muneaux, Yvette A.; Assens, Jean-Louis A.; et al.
Journal of Medicinal Chemistry, 1993 , vol. 36, # 22 p. 3371 - 3380
1: 96 percent / AcOH / xylene / 6.5 h / Heating 2: 1.) NaH / 1.) DMF, RT, 0.5 h, 2.) DMF, RT, 1 h View Scheme
参考文献
Bernhart, Claude A.; Perreaut, Pierre M.; Ferrari, Bernard P.; Muneaux, Yvette A.; Assens, Jean-Louis A.; et al.
Journal of Medicinal Chemistry, 1993 , vol. 36, # 22 p. 3371 - 3380
Bernhart, Claude A.; Perreaut, Pierre M.; Ferrari, Bernard P.; Muneaux, Yvette A.; Assens, Jean-Louis A.; et al.
Journal of Medicinal Chemistry, 1993 , vol. 36, # 22 p. 3371 - 3380