1: palladium dichloride; potassium carbonate / acetone; water / 0.17 h / 110 °C / |Microwave irradiation 2: palladium 10 on activated carbon; hydrogenchloride; hydrogen / water; methanol / 24 h / 2585.81 Torr View Scheme
参考文献
Mosberg, Henry I.; Yeomans, Larisa; Harland, Aubrie A.; Bender, Aaron M.; Sobczyk-Kojiro, Katarzyna; Anand, Jessica P.; Clark, Mary J.; Jutkiewicz, Emily M.; Traynor, John R.
Journal of Medicinal Chemistry, 2013 , vol. 56, # 5 p. 2139 - 2149