De Belin, Jackie Y; Romero-Martin, Maria-Rosario; Finn, Paul W; Sayers, Lee G; Law, Norman M; Billington, David C; Ryley, Stephen; Bhattacharya, Shoumo
Patent: US2003/229108 A1, 2003 ;
Location in patent: Page 37 ;
1: With 3-methyl-2-amino-pyridine; Wilkinson's catalyst; α,α,α-Trifluoro-p-toluic acid; cyclohexylamine in toluene
T=130°C; 12 h;
2: With hydrogenchloride; water in tetrahydrofuran
参考文献
Cha, Kyung-Mi; Lee, Hyejeong; Park, Jung-Woo; Lee, Yura; Jo, Eun-Ae; Jun, Chul-Ho
Chemistry - An Asian Journal, 2011 , vol. 6, # 8 p. 1926 - 1930