反应条件
1.1: acetic acid / 1 h / 100 °C
2.1: AlCl3, aluminium chloride / 1,2-dichloro-ethane / 0.5 h / 0 °C
2.2: 2 h / 0 - 20 °C
View Scheme
参考文献
PRESIDENT AND FELLOWS OF HARVARD COLLEGE; FINLEY, Daniel; KING, Randall, W.; LEE, Byung-Hoon; LEE, Min, Jae; GAHMAN, Timothy, C.
Patent: WO2011/94545 A2, 2011 ;
WO 2011/094545 A1