一氯乙醛合成路线

参考文献

Shao, Linjun; Xing, Guiying; He, Luyao; Chen, Ji; Xie, Hangqing; Liang, Xuezheng; Qi, Chenze
Applied Catalysis A: General, 2012 , vol. 443-444, p. 133 - 137

5049-61-6氨基吡嗪+

107-20-0一氯乙醛

274-79-3吲哚[1,2-A]吡嗪

参考文献

JIANGSU HANSOH PHARMACEUTICAL CO., LTD.; Tang, Peng Cho; Li, Xin; Li, Xiangqin; Chen, Yang; Wang, Bin; Zhu, Zhe
Patent: US2013/131068 A1, 2013 ;
Location in patent: Paragraph 0115; 0116 ;

107-20-0一氯乙醛+

98651-70-82-氨基-4-甲氧基烟腈

834869-04-47-甲氧基咪唑并[1,2-a]吡啶-8-甲腈

参考文献

ARENA PHARMACEUTICALS INC.
Patent: WO2009/23253 A2, 2009 ;
Location in patent: Page/Page column 77 ;
WO 2009/023253 A2

695-34-12-氨基-4-甲基吡啶+

107-20-0一氯乙醛

874-39-57-甲基咪唑并[1,2-A]砒啶

参考文献

Journal of Medicinal Chemistry, , vol. 35, # 23 p. 4415 - 4424

107-20-0一氯乙醛+

6937-03-72-氨基异烟酸甲酯

86718-01-6咪唑并[1,2-a]吡啶-7-羧酸甲酯

参考文献

ASTEX THERAPEUTICS LIMITED
Patent: WO2009/47506 A1, 2009 ;
Location in patent: Page/Page column 101; 107 ;
WO 2009/047506 A1

1824-81-32-氨基-6-甲基吡啶+

107-20-0一氯乙醛

933-69-75-甲基咪唑并[1,2-a]吡啶

参考文献

Ikemoto, Tomomi; Wakimasu, Mitsuhiro
Heterocycles, 2001 , vol. 55, # 1 p. 99 - 108

107-20-0一氯乙醛+

13534-99-12-氨基-3-溴吡啶

850349-02-9

参考文献

Bischoff, Francois; Berthelot, Didier; De Cleyn, Michel; MacDonald, Gregor; Minne, Garrett; Oehlrich, Daniel; Pieters, Serge; Surkyn, Michel; Trabanco, Andres A.; Tresadern, Gary; Van Brandt, Sven; Velter, Ingrid; Zaja, Mirko; Borghys, Herman; Masungi, Chantal; Mercken, Marc; Gijsen, Harrie J. M.
Journal of Medicinal Chemistry, 2012 , vol. 55, # 21 p. 9089 - 9106,18

107-20-0一氯乙醛+

446273-59-2

933190-51-3

参考文献

CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO); SNODIN, Michael D; PASTOR FERNANDEZ, Joaquín; MARTÍNEZ GONZÁLEZ, Sonia; BLANCO-APARICIO, Carmen; LORENZO GARCÍA, Milagros; RAMOS LIMA, Francisco Javier
Patent: WO2013/5041 A1, 2013 ;
Location in patent: Page/Page column 71 ;
WO 2013/005041 A1

参考文献

Pastor-Fernández, Joaquin; Bartolomé-Nebreda, José Manuel; Macdonald, Gregor James; Conde-Ceide, Susana; Delgado-González, Óscar; Vanhoof, Greta Constantia Peter; Van Gool, Michiel Luc Maria; Martin-Martín, María Luz; Alonso-de Diego, Sergio-Alvar; Swinney, Kelly Ann; Leys, Carina; Weerts, Johan Erwin Edmond; Wuyts, Stijn
Patent: US2011/269752 A1, 2011 ;
Location in patent: Page/Page column 29 ;

107-20-0一氯乙醛+

1072-98-62-氨基-5-氯吡啶

885275-59-2

参考文献

Buckley, George M.; Fosbeary, Richard; Fraser, Joanne L.; Gowers, Lewis; Higueruelo, Alicia P.; James, Lynwen A.; Jenkins, Kerry; Mack, Stephen R.; Morgan, Trevor; Parry, David M.; Pitt, William R.; Rausch, Oliver; Richard, Marianna D.; Sabin, Verity
Bioorganic and Medicinal Chemistry Letters, 2008 , vol. 18, # 12 p. 3656 - 3660