反应条件
1: 40 percent / pyridine / diethyl ether; H2O / 1.) 0 deg C, 30 min, 2.) reflux, 4 h
2: 62.6 percent / Ag2CO3 / propan-2-ol; CHCl3; dimethylformamide; H2O / 6 h / 65 °C
View Scheme
参考文献
Meyer, Karen L.; Marasco, Canio J.; Morris-Natschke, Susan L.; Ishaq, Khalid S.; Piantadosi, Claude; Kucera, Louis S.
Journal of Medicinal Chemistry, 1991 , vol. 34, # 4 p. 1377 - 1383