1: With ammonia in diethyl ether T=0°C; 2: With pyridine; acetic anhydride 1 h; Heating / reflux; 3: With sodium tetrahydroborate in methanol
参考文献
ZAPAQ, INC.; THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ILLINOIS; OKLAHOMA MEDICAL RESEARCH FOUNDATION
Patent: WO2006/34277 A1, 2006 ;
Location in patent: Page/Page column 63 ;
WO 2006/034277 A1
Abbott, Shaun D.; Lane-Bell, Patricia; Sidhu, Kanwar P. S.; Vederas, John C.
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