1: piperidine; formaldehyd in ethanol; water Mannich Aminomethylation; 0.5 h; 2: 3-Hydroxy-2(1H)-pyridinone in ethanol; water T=45°C; Mannich Aminomethylation; 12 h;
参考文献
Xie, Wen Lin; Xiao, Chuang Ping; Xie, Ling; Zhou, Ying; Li, Xue Feng; Tang, Xu Fu; Yuan, Chun Tao; Qiu, Ming Hua
Research on Chemical Intermediates, 2012 , vol. 38, # 7 p. 1699 - 1705