1-甲基吡唑-5-甲酸合成路线

参考文献

Galapagos NV
Patent: WO2009/71706 A1, 2009 ;
Location in patent: Page/Page column 48 ;
WO 2009/071706 A1

1621-91-6吡唑-3-甲酸+

77-78-1硫酸二甲酯

16034-46-11-甲基吡唑-5-甲酸+

25016-20-01-甲基吡唑-3-甲酸

参考文献

J. Gen. Chem. USSR (Engl. Transl.), , vol. 52, # 11 p. 2592 - 2598,2291 - 2296

930-36-9N-甲基吡唑+

201230-82-2

16034-46-11-甲基吡唑-5-甲酸

参考文献

Takeda Pharmaceutical Company Limited
Patent: EP2530078 A1, 2012 ;
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694-31-51,5-二甲基吡唑

16034-46-11-甲基吡唑-5-甲酸

参考文献

Manaev, Yu. A.; Andreeva, M. A.; Perevalov, V. P.; Stepanov, B. I.; Dubrovskaya, V. A.; Seraya, V. I.
J. Gen. Chem. USSR (Engl. Transl.), 1982 , vol. 52, # 11 p. 2592 - 2598,2291 - 2296

930-36-9N-甲基吡唑

16034-46-11-甲基吡唑-5-甲酸

参考文献

Journal of the American Chemical Society, , vol. 80, p. 6271,6273

Justus Liebigs Annalen der Chemie, , vol. 625, p. 55,60

27258-33-91-甲基-1H-吡唑-5-甲醛

16034-46-11-甲基吡唑-5-甲酸

参考文献

Lyalin; Petrosyan
Russian Chemical Bulletin, 2012 , vol. 61, # 6 p. 1148 - 1153
Izv. Akad. Nauk, Ser. Khim., 2012 , vol. 61, # 6 p. 1139 - 1143,5

930-36-9N-甲基吡唑+

109-72-8正丁基锂+

60-29-7乙醚

16034-46-11-甲基吡唑-5-甲酸

参考文献

Journal of the American Chemical Society, , vol. 80, p. 6271,6273

Justus Liebigs Annalen der Chemie, , vol. 625, p. 55,60

930-36-9N-甲基吡唑+

60-29-7乙醚+

591-51-5苯基锂

16034-46-11-甲基吡唑-5-甲酸

参考文献

Journal of the American Chemical Society, , vol. 80, p. 6271,6273

Justus Liebigs Annalen der Chemie, , vol. 625, p. 55,60

16034-46-11-甲基吡唑-5-甲酸

92534-69-51-甲基-4-硝基-1H-吡唑-5-羧酸

参考文献

Perevalov, V. P.; Andreeva, M. A.; Manaev, Yu. A.; Isaev, Sh. G.; Baryshnenkova, L. I.; Stepanov, B. I.
Journal of Organic Chemistry USSR (English Translation), 1984 , vol. 20, # 5 p. 976 - 980
Zhurnal Organicheskoi Khimii, 1984 , vol. 20, # 5 p. 1073 - 1078

16034-46-11-甲基吡唑-5-甲酸

92534-73-14-氨基-1-甲基-1H-吡唑-5-甲酰胺

参考文献

Lee, Wendy; Ortwine, Daniel F.; Bergeron, Philippe; Lau, Kevin; Lin, Lichuan; Malek, Shiva; Nonomiya, Jim; Pei, Zhonghua; Robarge, Kirk D.; Schmidt, Stephen; Sideris, Steve; Lyssikatos, Joseph P.
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