4-溴-2-甲基-2H-1,2,3-三唑合成路线 (共 3 条)
反应条件
n-butyllithium in tetrahydrofuran T=-78°C;
参考文献
CONSTELLATION PHARMACEUTICALS, INC.; ALBRECHT, Brian, K.; GEHLING, Victor, S.; HEWITT, Michael, C.; TAYLOR, Alexander, M.; HARMANGE, Jean-Christophe
Patent: WO2012/151512 A2, 2012 ;
Location in patent: Page/Page column 151 ;
参考文献
Pedersen
Acta Chemica Scandinavica (1947-1973), 1959 , vol. 13, p. 888,890
参考文献
Pedersen
Acta Chemica Scandinavica (1947-1973), 1959 , vol. 13, p. 888,890