反应条件
1: With potassium carbonate; N-fluoro-N-(phenylsulfonyl)benzene-sulfonamide in N,N-dimethyl-formamide; acetonitrile
T=-15°C;
2: With hydrogenchloride in dichloromethane; N,N-dimethyl-formamide; acetonitrile
T=20°C; 2 h;
参考文献
Verniest, Guido; Van Hende, Eva; Surmont, Riccardo; De Kimpe, Norbert
Organic Letters, 2006 , vol. 8, # 21 p. 4767 - 4770