1: With n-butyllithium in tetrahydrofuran T=-78°C; 2 h; 2: With boric acid trimethyl ester in tetrahydrofuran T=-78 - 20°C; 19 h; 3: With hydrogenchloride in tetrahydrofuran; water T=20°C;
参考文献
STERIX LIMITED
Patent: WO2007/96647 A2, 2007 ;
Location in patent: Page/Page column 125-126 ;
WO 2007/096647 A2