反应条件
1: in N,N-dimethyl acetamide T=60 - 70°C; 24 h; 2: With sodium hydrogencarbonate in N,N-dimethyl acetamide T=0°C;
参考文献
Homma, Akie; Sato, Haruhiko; Okamachi, Akira; Emura, Takashi; Ishizawa, Takenori; Kato, Tatsuya; Matsuura, Tetsu; Sato, Shigeo; Tamura, Tatsuya; Higuchi, Yoshinobu; Watanabe, Tomoyuki; Kitamura, Hidetomo; Asanuma, Kentaro; Yamazaki, Tadao; Ikemi, Masahisa; Kitagawa, Hironoshin; Morikawa, Tadashi; Ikeya, Hitoshi; Maeda, Kazuaki; Takahashi, Koichi; Nohmi, Kenji; Izutani, Noriyuki; Kanda, Makoto; Suzuki, Ryochi
Bioorganic and Medicinal Chemistry, 2009 , vol. 17, # 13 p. 4647 - 4656