反应条件
1: 69 percent / pyridine / 24 h / Ambient temperature 2: 80 percent / acetonitrile / Ambient temperature 3: 1) AIBN, n-Bu3SnH, 2) aq.AcOH / 1) toluene, 110-120 deg C, 3.5 h, 2) 50 deg C, 30 min View Scheme
参考文献
Journal of Medicinal Chemistry, , vol. 32, # 5 p. 1135 - 1140