1: With benzotriazol-1-ol; 1-ethyl-(3-(3-dimethylamino)propyl)-carbodiimide hydrochloride in acetonitrile 0.0833333 h; Inert atmosphere; 2: With triethylamine in acetonitrile 1.5 h; Inert atmosphere;
参考文献
Hyster, Todd K.; Rovis, Tomislav
Journal of the American Chemical Society, 2010 , vol. 132, # 30 p. 10565 - 10569