Stout, David M.; Matier, W. L.; Barcelon-Yang, Cynthia; Reynolds, Robert D.; Brown, Barry S.
Journal of Medicinal Chemistry, 1984 , vol. 27, # 10 p. 1347 - 1350
1: With aluminium trichloride
T=20°C; Acylation; demethylation; ethylation; 22 h;
2: With piperidine in water
Cyclization; 47 h; Heating;
参考文献
Fernandes, Eduarda G. R.; Silva, Artur M. S.; Cavaleiro, Jose A. S.; Silva, Francisco M.; Borges, M. Fernanda M.; Pinto, Madalena M. M.
Magnetic Resonance in Chemistry, 1998 , vol. 36, # 4 p. 305 - 309