1: CH2Cl2 / 2 h / 20 °C 2: thionyl chloride / 1 h / 25 °C 3: tetrahydrofuran / 2 h / 20 °C 4: 88 percent / 4.5 N aq. HCl / 12 h / Heating View Scheme
参考文献
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Journal of Medicinal Chemistry, 1991 , vol. 34, # 8 p. 2525 - 2547
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Thompson
Journal of the American Chemical Society, 1937 , vol. 59, p. 816