1,2,3-噻唑(1,5-a)吡啶合成路线 （共 26 条）
反应条件
palladium diacetate; caesium carbonate; triphenylphosphine T=140°C; 72 h; Inert atmosphere;
参考文献
Arkivoc, , vol. 2012, # 9 p. 229 - 241
反应条件
1: n-butyllithium / tetrahydrofuran / -40 °C 2: 4.2 percent / styrylazide / -78 °C View Scheme
参考文献
Abarca; Asensio; Jones; Mouat
Tetrahedron, 1989 , vol. 45, # 22 p. 7041 - 7048
反应条件
sulfuric acid in water T=95°C; 5 h;
参考文献
Journal of the Chemical Society, Perkin Transactions 1: Organic and Bio-Organic Chemistry (1972-1999), , p. 2719 - 2724
反应条件
palladium 10 on activated carbon; zinc in ethanol; water T=150°C; 24 h; Autoclave;
参考文献
Arkivoc, , vol. 2014, # 2 p. 175 - 186
反应条件
selenium(IV) oxide in chlorobenzene T=132°C; 6 h;
参考文献
Jones, Gurnos; Mouat, Deborah J.; Tonkinson, Daryl J.
Journal of the Chemical Society, Perkin Transactions 1: Organic and Bio-Organic Chemistry (1972-1999), 1985 , p. 2719 - 2724
反应条件
palladium diacetate; caesium carbonate; triphenylphosphine in N,N-dimethyl-formamide T=160°C; 24 h; Inert atmosphere;
参考文献
Arkivoc, , vol. 2012, # 9 p. 229 - 241
反应条件
palladium diacetate; caesium carbonate; triphenylphosphine T=140°C; 72 h; Inert atmosphere;
参考文献
Arkivoc, , vol. 2012, # 9 p. 229 - 241
反应条件
n-butyllithium; diisopropylamine
1.) ether, hexane, -40 deg C, 6 h, 2.) ether, hexane, RT, overnight; Yield given. Multistep reaction;
参考文献
Latham, Elliot J.; Stanforth, Stephen P.
Journal of Heterocyclic Chemistry, 1995 , vol. 32, # 3 p. 787 - 790
反应条件
acetic acid
T=118°C; 2 h;
参考文献
Jones, Gurnos; Mouat, Deborah J.; Tonkinson, Daryl J.
Journal of the Chemical Society, Perkin Transactions 1: Organic and Bio-Organic Chemistry (1972-1999), 1985 , p. 2719 - 2724
参考文献
Boyer; Wolford
Journal of the American Chemical Society, 1958 , vol. 80, p. 2741
