反应条件
1: 1H-tetrazole With sodium hydride in N,N-dimethyl-formamide T=20°C; 1.5 h; 2: 1-bromo-3-chloro-propane in N,N-dimethyl-formamide T=20°C;
参考文献
SUNSHINE LAKE PHARMA CO., LTD.; ZHANG, Yingjun; ZHANG, Jiancun; WANG, Xiaojun; LIN, Runfeng; CAO, Shengtian; WANG, Zhaohe; LI, Jing
Patent: WO2014/12360 A1, 2014 ;
Location in patent: Paragraph 00408 ;