1,2,3,4-四氢-2-萘胺合成路线 (共 39 条)
反应条件
supported Candida antartica lipase B in tert-butyl methyl ether T=38 - 40°C; 20 h; Molecular sieveEnzymatic reaction; optical yield given as percent eeenantioselective reaction;
参考文献
Poulhes, Florent; Vanthuyne, Nicolas; Bertrand, Michele P.; Gastaldi, Stephane; Gil, Gerard
Journal of Organic Chemistry, 2011 , vol. 76, # 17 p. 7281 - 7286
反应条件
coated protease in 3-methyl pentan-3-ol T=21°C; 144 h; Resolution of racemateEnzymatic reaction; enantioselective reaction;
参考文献
Queyroy, Severine; Vanthuyne, Nicolas; Gastaldi, Stephane; Bertrand, Michele P.; Gil, Gerard
Advanced Synthesis and Catalysis, 2012 , vol. 354, # 9 p. 1759 - 1764
反应条件
formic acid
4 h; Heating;
参考文献
Bucholtz, Ehren C.; Brown, Randal L.; Tropsha, Alexander; Booth, Raymond G.; Wyrick, Steven D.
Journal of Medicinal Chemistry, 1999 , vol. 42, # 16 p. 3041 - 3054
反应条件
1: water; formic acid
2: water; formic acid
View Scheme
参考文献
Cymerman Craig et al.
Australian Journal of Chemistry, 1959 , vol. 12, p. 447,450,451
参考文献
Chiavarelli et al.
Rend.Ist.super.Sanita, 1952 , vol. 15, p. 862,865
参考文献
Bamberger; Kitschelt
Chemische Berichte, 1890 , vol. 23, p. 885
参考文献
Bamberger; Kitschelt
Chemische Berichte, 1890 , vol. 23, p. 885
参考文献
Bamberger; Mueller
Chemische Berichte, 1888 , vol. 21, p. 1116
参考文献
Bamberger; Mueller
Chemische Berichte, 1888 , vol. 21, p. 1116