1.1: CH2Cl2 / 16 h / 20 °C 2.1: NaH / tetrahydrofuran / 3 h / 65 °C 2.2: 81 percent / tetrahydrofuran / 18 h / 65 °C 3.1: 72 percent / KOH / methanol; H2O / 18 h / 80 °C View Scheme
参考文献
Adam, Waldemar; Pastor, Aurelia; Wirth, Thomas
Organic Letters, 2000 , vol. 2, # 9 p. 1295 - 1297