1: With potassium phosphate; tetrakis(triphenylphosphine) palladium(0) in DMF (N,N-dimethyl-formamide); water
T=150°C; 0.5 h; Microwave irradiation;
2: With hydrogenchloride in DMF (N,N-dimethyl-formamide); water
参考文献
Carter, Percy H.; Cherney, Robert J.; Batt, Douglas G.; Brown, Gregory D.; Duncia, John V.; Gardner, Daniel S.; Yang, Michael G.
Patent: US2005/54626 A1, 2005 ;
Location in patent: Page/Page column 42 ;
US 20050054626 A1