反应条件
1.1: N-ethyl-N,N-diisopropylamine / dichloromethane / -5 - 30 °C / Inert atmosphere; Industry scale 2.1: sodium hydride / 1-methyl-pyrrolidin-2-one; mineral oil / -5 - 20 °C / Industry scale; Inert atmosphere 2.2: 20 - 55 °C / Industry scale; Inert atmosphere View Scheme
参考文献
Xu, Yaozu; Ogunsina, Makanjuola; Samadder, Pranati; Arthur, Gilbert; Schweizer, Frank
ChemMedChem, 2013 , vol. 8, # 3 p. 511 - 520