1: acetyl chloride With pyridine in 1-methyl-pyrrolidin-2-one
T=20°C;
2: 2-Pyridinylmethylamine in tetrahydrofuran
T=20°C; Further stages.;
参考文献
Chang, Young-Tae; Choi, Jaehwa; Ding, Sheng; Prieschl, Eva E.; Baumruker, Thomas; Lee, Jae-Mok; Chung, Sung-Kee; Schultz, Peter G.
Journal of the American Chemical Society, 2002 , vol. 124, # 9 p. 1856 - 1857