反应条件
sodium methylate; caesium carbonate; potassium iodide; Merrifield resin; (1,1'-bis(diphenylphosphino)ferrocene)palladium(II) dichloride 1.) DMF, 80 deg C, 18 h; 2.) THF, r.t., 18 h; 3.) THF, 70 deg C, 18 h; Yield given. Multistep reaction;
参考文献
Marquais, Sophie; Arlt, Michael
Tetrahedron Letters, 1996 , vol. 37, # 31 p. 5491 - 5494