反应条件
1: ethanol / 2 h / Reflux
2: 4-(N,N-dimethlyamino)pyridine; 1-ethyl-(3-(3-dimethylamino)propyl)-carbodiimide hydrochloride / chloroform / 24 h
3: sodium hydroxide / 1,4-dioxane / 2.5 h / 60 °C
View Scheme
参考文献
Xu, Qinyuan; Huang, Li; Liu, Juan; Ma, Liang; Chen, Tao; Chen, Jinying; Peng, Fei; Cao, Dong; Yang, Zhuang; Qiu, Neng; Qiu, Jingxiang; Wang, Guangcheng; Liang, Xiaolin; Peng, Aihua; Xiang, Mingli; Wei, Yuquan; Chen, Lijuan
European Journal of Medicinal Chemistry, 2012 , vol. 52, p. 70 - 81