1: With N,N-dimethyl-formamide; trichlorophosphate T=0 - 45°C; 1.5 h; 2: With ammonia in water T=0 - 10°C; 1 h;
参考文献
Ruck, Rebecca T.; Huffman, Mark A.; Stewart, Gavin W.; Cleator, Ed; Kandur, Wynne V.; Kim, Mary M.; Zhao, Dalian
Organic Process Research and Development, 2012 , vol. 16, # 8 p. 1329 - 1337