反应条件
1: hydroxylamine hydrochloride With sodium hydrogencarbonate in 1,4-dioxane; water T=0 - 5°C; 0.666667 h; 2: chlorodiphenylphosphine oxide in 1,4-dioxane; water T=0 - 20°C; 2.5 h;
参考文献
3-V BIOSCIENCES, INC.; OSLOB, Johan D.; MCDOWELL, Robert S.; JOHNSON, Russell; YANG, Hanbiao; EVANCHIK, Marc; ZAHARIA, Cristiana A.; CAI, Haiying; HU, Lily W.
Patent: WO2014/8197 A1, 2014 ;
Location in patent: Page/Page column 134; 135 ;