potassium hydroxide in dimethyl sulfoxide T=20°C; 1 h;
参考文献
Albers, Harald M. H. G.; Hendrickx, Loes J. D.; Van Tol, Rob J. P.; Hausmann, Jens; Perrakis, Anastassis; Ovaa, Huib
Journal of Medicinal Chemistry, 2011 , vol. 54, # 13 p. 4619 - 4626
1: sodium azide / dimethyl sulfoxide / 1 h / 80 °C 2: triphenylphosphine / methanol / 1 h / |Reflux View Scheme
参考文献
DANA-FARBER CANCER INSTITUTE, INC.; THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA; THE UNITED STATES OF AMERICA as represented by THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVIECES; BRYN MAWR COLLEGE; THE JOHNS HOPKINS UNIVERSITY; THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK; SODROSKI, Joseph; LALONDE, Judith, M.; SMITH, Amos, B., iii; KWONG, Peter, D.; KWON, Young Do; JONES, David, M.; SUN, Alexander, W.; COURTER, Joel, R.; SOETA, Takahiro; KOBAYASHI, Toyoharu; PRINCIOTTO, Amy M.; WU, Xueling; MASCOLA, John R.; SCHON, Arne; FREIRE, Ernesto; MADANI, Navid; LE-KHAC, Matthew; HENDRICKSON, Wayne, A.
Patent: WO2013/90696 A1, 2013 ;
