反应条件
1: 1.) NaH / 1.) THF, DMF, 20 min, 2.) THF, DMF, 30 min
2: 1.) NaH / 1.) DMF, 15 min, 2.) DMF, THF, a.) 30 min, b.) RT, overnight
View Scheme
参考文献
Gu, Zi-Qiang; Wong, Garry; Dominguez, Celia; Costa, Brian R. de; Rice, Kenner C.; Skolnick, Phil
Journal of Medicinal Chemistry, 1993 , vol. 36, # 8 p. 1001 - 1006