1: 70 percent / K2CO3 / acetone / 1 h / Heating 2: 81 percent / 3-chloroperoxybenzoic acid / CH2Cl2 / 2.5 h / -10 °C 3: 68 percent / aq. perchloric acid / dioxane / 1 h / 20 °C View Scheme
参考文献
Bellevue III, Frank H.; Woster, Patrick M.; Edwards, David J.; He, Kan; Hollenberg, Paul F.
Bioorganic and Medicinal Chemistry Letters, 1997 , vol. 7, # 20 p. 2593 - 2598