反应条件
1: 1.) n-BuLi / 1.) Et2O, hexane, -70 deg C, 2.) Et2O, hexane, THF, -70 deg C, 1 h 2: 1.) (COCl)2, DMSO, 2.) Et3N / 1.) CH2Cl2, -70 deg C, 45 min, 2.) CH2Cl2, from -70 deg C to 25 deg C View Scheme
参考文献
Ackerley, Norman; Brewster, Andrew G.; Brown, George R.; Clarke, David S.; Foubister, Alan J.; et al.
Journal of Medicinal Chemistry, 1995 , vol. 38, # 10 p. 1608 - 1628