反应条件
1: 3-(1H pyrazol-3-yl)-pyridine With sodium hydride in N,N-dimethyl-formamide
T=20°C; 0.5 h;
2: methyl iodide in N,N-dimethyl-formamide
T=20°C; 3 h;
参考文献
Del Giudice, Maria Rosaria; Mustazza, Carlo; Borioni, Anna; Gatta, Franco; Tayebati, Khosrow; Amenta, Francesco; Tucci, Paolo; Pieretti, Stefano
Archiv der Pharmazie, 2003 , vol. 336, # 3 p. 143 - 154