1: phenylacetic acid With 1,1'-carbonyldiimidazole in tetrahydrofuran Acylation; 2: malonic acid ethyl ester monopotassium salt With magnesium chloride in tetrahydrofuran Substitution; decarboxylation;
参考文献
Bioorganic and Medicinal Chemistry, , vol. 7, # 6 p. 991 - 1002