反应条件
1: lithium aluminium tetrahydride / tetrahydrofuran / 17.25 h / 0 °C / |Inert atmosphere; |Reflux 2: triethylamine / dichloromethane / 2 h / 0 - 20 °C 3: triethylamine; 4-(N,N-dimethlyamino)pyridine; p-toluenesulfonyl chloride / dichloromethane / 0 - 20 °C View Scheme
参考文献
Li, Meiling; Hawkins, Alison; Barber, David M.; Bultinck, Patrick; Herrebout, Wouter; Dixon, Darren J.
Chemical Communications, 2013 , vol. 49, # 46 p. 5265 - 5267