1: With acetic acid in dichloromethane
T=20°C; 1 h;
2: With sodium tris(acetoxy)borohydride in dichloromethane
T=0 - 20°C; 16 h;
3: With sodium hydroxide in dichloromethane; water
0.5 h;
参考文献
GLAXO GROUP LIMITED
Patent: WO2004/56369 A1, 2004 ;
Location in patent: Page/Page column 47-48 ;