联硼酸频那醇酯合成路线

Burger, Matthew T.; Pecchi, Sabina; Wagman, Allan; Ni, Zhi-Jie; Knapp, Mark; Hendrickson, Thomas; Atallah, Gordana; Pfister, Keith; Zhang, Yanchen; Bartulis, Sarah; Frazier, Kelly; Ng, Simon; Smith, Aaron; Verhagen, Joelle; Haznedar, Joshua; Huh, Kay; Iwanowicz, Ed; Xin, Xiaohua; Menezes, Daniel; Merritt, Hanne; Lee, Isabelle; Wiesmann, Marion; Kaufman, Susan; Crawford, Kenneth; Chin, Michael; Bussiere, Dirksen; Shoemaker, Kevin; Zaror, Isabel; Maira, Sauveur-Michel; Voliva, Charles F.
ACS Medicinal Chemistry Letters, 2011 , vol. 2, # 10 p. 774 - 779

944401-56-32-氨基-5-溴-4-三氟甲基吡啶+

73183-34-3联硼酸频那醇酯

944401-57-42-氨基-4-三氟甲基-5-吡啶硼酸哪醇酯

参考文献

UNIVERSITY OF BASEL; CMILJANOVIC, Vladimir; CMILJANOVIC, Natasa; GIESE, Bernd; WYMANN, Matthias
Patent: WO2010/52569 A2, 2010 ;
Location in patent: Page/Page column 221-222 ;
WO 2010/052569 A2

1021919-24-34-溴-3-甲基-1H-吡唑-1-羧酸叔丁酯+

73183-34-3联硼酸频那醇酯

936250-20-3

参考文献

SIGNAL PHARMACEUTICALS, LLC
Patent: WO2008/51493 A2, 2008 ;
Location in patent: Page/Page column 181 ;

1453-58-3+

73183-34-3联硼酸频那醇酯

936250-20-3

参考文献

Larsen, Matthew A.; Hartwig, John F.
Journal of the American Chemical Society, 2014 , vol. 136, # 11 p. 4287 - 4299

73583-37-6+

73183-34-3联硼酸频那醇酯

458532-84-8

参考文献

Wang, Lianhui; Cui, Xiuling; Li, Jingya; Wu, Yusheng; Zhu, Zhiwu; Wu, Yangjie
European Journal of Organic Chemistry, 2012 , # 3 p. 595 - 603