反应条件
1: 6-chloro-2H-3,1-benzoxazine-2,4(1H)-dione With sodium hydride in N,N-dimethyl-formamide T=20°C; 1 h; 2: methyl bromide in N,N-dimethyl-formamide 18 h;
参考文献
Clark, Rachel L.; Clements, Carol J.; Barrett, Michael P.; MacKay, Simon P.; Rathnam, Rajendra P.; Owusu-Dapaah, George; Spencer, John; Huggan, Judith K.
Bioorganic and Medicinal Chemistry, 2012 , vol. 20, # 20 p. 6019 - 6033