1: 12 h; Inert atmosphereReflux; 2: With potassium oxide
参考文献
KOREA INSTITUTE OF SCIENCE AND TECHNOLOGY; YOO, Bok Ryul; HAN, Joon Soo; YOO, Jang Hyun
Patent: WO2011/81277 A2, 2011 ;
Location in patent: Page/Page column 12-13 ;
in acetonitrile T=120°C; 0.333333 h; microwave irradiation;
参考文献
Semple, Graeme; Skinner, Philip J.; Cherrier, Martin C.; Webb, Peter J.; Sage, Carleton R.; Tamura, Susan Y.; Chen, Ruoping; Richman, Jeremy G.; Connolly, Daniel T.
Journal of Medicinal Chemistry, 2006 , vol. 49, # 4 p. 1227 - 1230