反应条件
1: 3-keto-2H,3H-1,2-benzisothiazole 1,1-dioxide / dichloromethane / |Reflux; |Inert atmosphere
2: cesium fluoride / N,N-dimethyl-formamide / 24 h / 140 °C / 760.05 Torr
View Scheme
参考文献
Mita, Tsuyoshi; Higuchi, Yuki; Sato, Yoshihiro
Organic Letters, 2014 , vol. 16, # 1 p. 14 - 17