3-(1H-四唑-1-基)丙酸合成路线 （共 4 条）
反应条件
1: With triethylamine in acetonitrile
T=20°C; 24 h;
2: With hydrogenchloride in water
pH=1; Cooling with iceInert atmosphere;
参考文献
Nguyen-Trung, Anh Thu; Tritsch, Denis; Grosdemange-Billiard, Catherine; Rohmer, Michel
Bioorganic and Medicinal Chemistry Letters, 2013 , vol. 23, # 6 p. 1643 - 1647
反应条件
pyridine; 1H-tetrazole in water; isopropyl alcohol
参考文献
Ciba-Geigy Corporation
Patent: US4794109 A1, 1988 ;
反应条件
sodium azide in acetic acid
T=100°C; 3 h;
参考文献
Gaponik, P. N.; Karavai, V. P.; Grigor'ev, Yu. V.
Chemistry of Heterocyclic Compounds (New York, NY, United States), 1985 , vol. 21, # 11 p. 1255 - 1258
Khimiya Geterotsiklicheskikh Soedinenii, 1985 , vol. 21, # 11 p. 1521 - 1524
反应条件
N-benzyl-trimethylammonium hydroxide
参考文献
Wiley et al.
Journal of the American Chemical Society, 1955 , vol. 77, p. 2572
