反应条件
1: thionyl chloride / Reflux 2: nitric acid; tin(IV) chloride / dichloromethane / -70 °C 3: hydrogen / methanol / 20 °C 4: sodium methylate / methanol; N,N-dimethyl-formamide / 110 °C 5: trichlorophosphate / Reflux View Scheme
参考文献
Garofalo, Antonio; Goossens, Laurence; Baldeyrou, Brigitte; Lemoine, Amelie; Ravez, Severine; Six, Perrine; David-Cordonnier, Marie-Helene; Bonte, Jean-Paul; Depreux, Patrick; Lansiaux, Amelie; Goossens, Jean-Francois
Journal of Medicinal Chemistry, 2010 , vol. 53, # 22 p. 8089 - 8103