反应条件
1: 91 percent / pyridine, 4-dimethylaminopyridine / CH2Cl2 / Ambient temperature 2: 87 percent / pyridine, 4-dimethylaminopyridine / CH2Cl2 / Ambient temperature 3: phosphor buffer / lipase enzyme View Scheme
参考文献
Oberhauser, Th.; Bodenteich, M.; Faber, K.; Penn, G.; Griengl, H.
Tetrahedron, 1987 , vol. 43, # 17 p. 3931 - 3944