反应条件
1: 1.) NH3(gas), 2.) Na, 4.) TFA, 5.) NaOH 2: 68.7 percent / aq. Na2CO3 / dioxane / 3 h View Scheme
参考文献
Pearson, Daniel A.; Lister-James, John; McBride, William J.; Wilson, David M.; Martel, Lawrence J.; Civitello, Edgar R.; Taylor, John E.; Moyer, Brian R.; Dean, Richard T.
Journal of Medicinal Chemistry, 1996 , vol. 39, # 7 p. 1361 - 1371